SCHEMBL23175682

SCHEMBL23175682

O=C(c1ccc(Cl)cc1F)C1CC1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.55
CPS1 P31327 1/20 0.46
MGLL Q99685 4/20 0.44
CNR2 P34972 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 2/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP11B2 P19099 1/20 0.41
ACKR3 P25106 1/20 0.41
HSD11B1 P28845 2/20 0.40
TSHR P16473 1/20 0.40
CASP1 P29466 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL717212 0.93 KMT2A (0.49) KMT2ACPS1MGLLCNR2L3MBTL1
Hydrochloric Acid SCHEMBL15566650 0.89 KMT2A (0.46) KMT2ACPS1MGLLCNR2MEN1
SCHEMBL10395236 0.84 CPS1 (0.55) KMT2ACPS1MGLLMEN1ALDH1A1
SCHEMBL6141006 0.81 L3MBTL1 (0.61) KMT2ACPS1L3MBTL1MEN1ALDH1A1
SCHEMBL6141378 0.81 TSHR (0.57) KMT2AL3MBTL1MEN1ALDH1A1CYP1A2
SCHEMBL21381592 0.81 CPS1 (0.44) KMT2ACPS1MGLLL3MBTL1MEN1
SCHEMBL2304821 0.80 ALDH1A1 (0.51) KMT2ACPS1MGLLL3MBTL1MEN1
SCHEMBL11262337 0.79 ALDH1A1 (0.56) KMT2AMGLLMEN1ALDH1A1
SCHEMBL9267287 0.79 ABL1 (0.53) KMT2AMGLLMEN1ALDH1A1CYP1A2
SCHEMBL13398 0.79 CPS1 (0.46) KMT2ACPS1MGLLL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117177970-A Polycyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-05 CN disclosed
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed
WO-2021057890-A1 2H-BENZOPYRAN DERIVATIVES AS CRAC INHIBITORS 南京明德新药研发有限公司 2021-04-01 WO disclosed