SCHEMBL13398

SCHEMBL13398

Bc1ccc(C(=O)C2CC2)c(F)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CPS1 P31327 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.43
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 3/20 0.38
MAPT P10636 1/20 0.38
NPY2R P49146 1/20 0.38
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
NPC1 O15118 1/20 0.35
HSD11B1 P28845 3/20 0.34
PARP15 Q460N3 1/20 0.33
PARP10 Q53GL7 1/20 0.33
HTR1F P30939 1/20 0.33
DGAT1 O75907 1/20 0.33
MGLL Q99685 2/20 0.33
PDK2 Q15119 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17680658 0.86 HTR1F (0.41) CPS1L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL6141006 0.81 L3MBTL1 (0.61) CPS1L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL2304821 0.80 ALDH1A1 (0.51) CPS1L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL23175682 0.79 KMT2A (0.55) CPS1L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL30833732 0.79 DGAT1 (0.58) CPS1L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL13427 0.79 DGAT1 (0.58) CPS1L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL9156406 0.76 GAA (0.49) CPS1L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL28026637 0.76 L3MBTL1 (0.55) CPS1L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL28026635 0.76 L3MBTL1 (0.55) CPS1L3MBTL1KMT2AMEN1ALDH1A1
SCHEMBL256756 0.75 CES2 (0.43) ALDH1A1MAPTCES2CES1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011044187-A1 IMINOTHIADIAZINE DIOXIDE COMPOUNDS AS BACE INHIBITORS, COMPOSITIONS, AND THEIR USE SCHERING CORPORATION (US) 2011-04-14 WO disclosed