SCHEMBL23178593

SCHEMBL23178593

COc1c(F)cc(CN2CCC(N)CC2)cc1F

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 4/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
DBH P09172 1/20 0.43
BCHE P06276 2/20 0.40
BACE1 P56817 2/20 0.40
ACHE P22303 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
DRD3 P35462 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23178957 0.86 ACHE (0.50) KDM4EALDH1A1MEN1KMT2ATDP1
SCHEMBL11533768 0.83 KDM4E (0.63) KDM4EALDH1A1MEN1KMT2ATDP1
SCHEMBL17967915 0.83 MEN1 (0.44) KDM4EALDH1A1MEN1KMT2ATDP1
SCHEMBL2821325 0.82 ALDH1A1 (0.42) KDM4EALDH1A1GAAHTT
SCHEMBL17946120 0.81 DRD4 (0.55) KDM4EALDH1A1TDP1POLBSMN1; SMN2
SCHEMBL30815930 0.81 DRD4 (0.55) KDM4EALDH1A1TDP1POLBSMN1; SMN2
SCHEMBL6939806 0.80 SIGMAR1 (0.49) KDM4EALDH1A1MEN1KMT2A
SCHEMBL1604858 0.77 SIGMAR1 (0.46) ALDH1A1MEN1KMT2AACHESMN1; SMN2
SCHEMBL8108284 0.77 SIGMAR1 (0.46) ALDH1A1MEN1KMT2AACHESMN1; SMN2
SCHEMBL3144826 0.76 ALDH1A1 (0.65) KDM4EALDH1A1DRD3HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574176-B Heteroaryl compound and application thereof 隆泰申医药科技(南京) 有限公司 2024-03-15 CN disclosed
WO-2021057696-A1 HETEROARYL COMPOUND AND APPLICATION THEREOF 隆泰申医药科技(南京)有限公司 2021-04-01 WO disclosed
CN-112574176-A Heteroaryl compound and application thereof 隆泰申医药科技(南京) 有限公司 2021-03-30 CN disclosed