SCHEMBL23197871

SCHEMBL23197871

C/C=C(/N=C(C)\C(C=N)=C(/C)Nc1cccc(SC)c1)NC1CCCC1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.43
MEN1 O00255 4/20 0.43
MAPT P10636 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
POLB P06746 2/20 0.39
RXFP1 Q9HBX9 2/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
PKM P14618 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 2/20 0.36
TP53 P04637 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HPGD P15428 1/20 0.35
ALOX12 P18054 1/20 0.35
NPC1 O15118 2/20 0.35
LMNA P02545 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23197827 0.73
SCHEMBL2751753 0.70 RAB9A (0.67) KMT2AMEN1MAPTCYP1A2CYP3A4
SCHEMBL7865726 0.62 MAPT (0.60) KMT2AMEN1MAPTCYP1A2CYP3A4
SCHEMBL23197819 0.61 MEN1 (0.33) KMT2AMEN1
SCHEMBL23197815 0.61 LMNA (0.41) KMT2AMEN1MAPTPOLBRXFP1
SCHEMBL27699157 0.61 MAPT (0.63) KMT2AMEN1MAPTCYP1A2CYP3A4
SCHEMBL7612008 0.60 KMT2A (0.60) KMT2AMEN1MAPTCYP1A2CYP3A4
SCHEMBL6716900 0.60 MAPT (0.62) KMT2AMEN1MAPTCYP1A2CYP3A4
SCHEMBL5208634 0.59 MAPT (0.70) KMT2AMEN1MAPTCYP1A2CYP3A4
SCHEMBL23198512 0.59 P2RX1 (0.40) MAPTPOLBALOX15TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021064077-A1 SUBSTITUTED PYRAZOLOPYRIMIDINES AS IRAK4 INHIBITORS BAYER AKTIENGESELLSCHAFT (DE) 2021-04-08 WO disclosed