SCHEMBL23212047

SCHEMBL23212047

Cn1cc(C2CCN(C(=O)O)CC2)c2cc(Cl)ccc21

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RORC P51449 14/20 0.50
DRD2 P14416 1/20 0.47
SLC6A4 P31645 1/20 0.47
KCNH2 Q12809 3/20 0.44
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17495546 0.85 RORC (0.50) RORCDRD2SLC6A4
SCHEMBL21382343 0.84 KCNH2 (0.52) DRD2SLC6A4KCNH2
SCHEMBL30568012 0.84 SCN9A (0.57) RORCKMT2A
SCHEMBL23212070 0.84 SCN9A (0.57) RORCKMT2A
SCHEMBL23211887 0.83 KCNH2 (0.44) DRD2SLC6A4KCNH2
SCHEMBL5705162 0.82 RORC (0.51) RORCKMT2A
SCHEMBL21385306 0.81 CNR1 (0.49) KCNH2
SCHEMBL22773323 0.81 SCN9A (0.43) RORCDRD2SLC6A4
SCHEMBL21382052 0.80 KCNH2 (0.46) DRD2SLC6A4KCNH2
SCHEMBL17495381 0.78 RORC (0.48) RORCDRD2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230117324-A1 OXAZINE MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS HOFFMANN-LA ROCHE INC. (US) 2023-04-20 US disclosed
EP-3768684-B1 OXAZINE MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS HOFFMANN LA ROCHE (CH) 2023-02-22 EP disclosed
US-20210107920-A1 OXAZINE MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS HOFFMANN-LA ROCHE INC. (US) 2021-04-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210107920-A1 OXAZINE MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS MGLL, LPL, LIPC RORC 2754/4885DRD2 3496/4885SLC6A4 4841/4885
US-20230117324-A1 OXAZINE MONOACYLGLYCEROL LIPASE (MAGL) INHIBITORS MGLL, LPL, LIPC RORC 2754/4885DRD2 3496/4885SLC6A4 4841/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.