SCHEMBL23213969

SCHEMBL23213969

CC(c1nccnc1-c1ccc(C(F)(F)F)cn1)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.35
MAOB P27338 1/20 0.34
SYK P43405 1/20 0.34
LMNA P02545 2/20 0.34
HIF1A Q16665 1/20 0.34
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
OGA O60502 1/20 0.33
TRPV3 Q8NET8 1/20 0.33
XPO1 O14980 1/20 0.33
ALDH1A1 P00352 1/20 0.33
UGCG Q16739 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
GALR3 O60755 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30010484 1.00 TRPV1 (0.35) TRPV1MAOBSYKLMNAHIF1A
SCHEMBL23212819 0.82 SMN1; SMN2 (0.37) LMNAALDH1A1ALOX15
SCHEMBL23212678 0.81 HPGD (0.41) MAOBL3MBTL1ALDH1A1
SCHEMBL29775963 0.81 HPGD (0.41) MAOBL3MBTL1ALDH1A1
SCHEMBL23212709 0.80 LMNA (0.42) LMNAHIF1AKDM4EALDH1A1
SCHEMBL23212691 0.80 LMNA (0.44) LMNAKDM4EL3MBTL1ALOX15
SCHEMBL24728835 0.78 ALOX15 (0.41) MAOBLMNAALDH1A1ALOX15
SCHEMBL31087595 0.78 ALOX15 (0.41) MAOBLMNAALDH1A1ALOX15
SCHEMBL31087599 0.78 ALOX15 (0.41) MAOBLMNAALDH1A1ALOX15
SCHEMBL24729152 0.78 ALOX15 (0.41) MAOBLMNAALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12583851-B2 Heteroaryl-substituted pyrazine derivatives as pesticides ELANCO ANIMAL HEALTH GMBH (DE) 2026-03-24 US disclosed
US-20230023326-A1 HETEROARYL-SUBSTITUTED PYRAZINE DERIVATIVES AS PESTICIDES ELANCO ANIMAL HEALTH GMBH (DE) 2023-01-26 US disclosed
EP-4041720-A1 HETEROARYL-SUBSTITUTED PYRAZINE DERIVATIVES AS PESTICIDES Bayer Animal Health GmbH (DE) 2022-08-17 EP disclosed
WO-2021069575-A1 HETEROARYL-SUBSTITUTED PYRAZINE DERIVATIVES AS PESTICIDES BAYER ANIMAL HEALTH GMBH (DE) 2021-04-15 WO disclosed
WO-2021069575-A1 HETEROARYL-SUBSTITUTED PYRAZINE DERIVATIVES AS PESTICIDES BAYER ANIMAL HEALTH GMBH (DE) 2021-04-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12583851-B2 Heteroaryl-substituted pyrazine derivatives as pesticides CBR3, CYCS, CWC15 TRPV1 2124/4885MAOB 4149/4885SYK 4515/4885
US-20230023326-A1 HETEROARYL-SUBSTITUTED PYRAZINE DERIVATIVES AS PESTICIDES DDT, PRXL2A, CAT TRPV1 2342/4885MAOB 1788/4885SYK 4201/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.