SCHEMBL23216816

SCHEMBL23216816

O=C(c1ccncc1)c1[c]ccc(Cl)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
LTA4H P09960 1/20 0.41
NAPRT Q6XQN6 1/20 0.38
TYK2 P29597 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
MAPK1 P28482 2/20 0.36
POLB P06746 1/20 0.36
ALDH1A1 P00352 1/20 0.36
JAK2 O60674 1/20 0.36
ENPP3 O14638 1/20 0.36
ALPL P05186 1/20 0.36
ENPP1 P22413 1/20 0.36
XIAP P98170 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MPO P05164 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16468436 0.75 LTA4H (0.47) LMNAKMT2AMEN1LTA4HNAPRT
SCHEMBL17188100 0.72 TSHR (0.42) MAPK1ALDH1A1SMN1; SMN2KDM4EHSD17B10
SCHEMBL28167045 0.71 ALDH1A1 (0.33) LMNAKMT2AL3MBTL1POLBALDH1A1
SCHEMBL29853983 0.69 MEN1 (0.46) LMNAKMT2AMEN1LTA4HNAPRT
SCHEMBL23215137 0.69 MEN1 (0.46) LMNAKMT2AMEN1LTA4HNAPRT
SCHEMBL725064 0.69 KMT2A (0.80) LMNAKMT2AMEN1LTA4HNAPRT
SCHEMBL23216806 0.68 JAK1 (0.44) LMNAKMT2AMEN1LTA4HNAPRT
SCHEMBL1969488 0.67 ALDH1A1 (0.39) KMT2AMEN1POLBALDH1A1ALPL
SCHEMBL5622548 0.67 ALPL (0.37) LMNAKMT2AMEN1ALDH1A1ALPL
SCHEMBL7452087 0.67 RAB9A (0.49) LMNAKMT2AMEN1LTA4HPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114727992-A Arylmethylene aromatic compounds as Kv1.3 potassium Shaker channel blockers D·E·萧尔研究有限责任公司 2022-07-08 CN disclosed
WO-2021071821-A1 ARYLMETHYLENE AROMATIC COMPOUNDS AS KV1.3 POTASSIUM SHAKER CHANNEL BLOCKERS D.E. SHAW RESEARCH, LLC (US) 2021-04-15 WO disclosed