SCHEMBL2330442

SCHEMBL2330442

Cc1cc([C@@H](C)NC(=O)c2cccc3ccc(C(C)(C)C(F)(F)F)nc23)c(Cl)cc1O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PDE2A O00408 2/20 0.35
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
POLB P06746 1/20 0.34
HSP90AA1 P07900 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CCR1 P32246 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2329497 0.91 CYP1A2 (0.39) CYP1A2CYP3A4CYP2C19TDP1KMT2A
SCHEMBL2328729 0.91 CYP1A2 (0.39) CYP1A2CYP3A4CYP2C19TDP1KMT2A
SCHEMBL2332508 0.90 MEN1 (0.41) PDE2AKMT2AMEN1POLBNPC1
SCHEMBL2106773 0.81 MEN1 (0.39) CYP1A2CYP2C19TDP1PDE2AKMT2A
SCHEMBL2329485 0.80 MEN1 (0.43) KMT2AMEN1POLBNPC1RAB9A
SCHEMBL2332116 0.80 MEN1 (0.43) KMT2AMEN1POLBNPC1RAB9A
SCHEMBL2326235 0.80 ADORA2A (0.34) PDE2A
SCHEMBL1841391 0.79 CCR1 (0.39) KMT2AMEN1RAB9ACCR1
SCHEMBL2332522 0.79 KMT2A (0.42) CYP1A2CYP3A4CYP2C19KMT2AMEN1
SCHEMBL1842345 0.79 ROCK2 (0.35) KMT2AMEN1CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222631-B1 SUBSTITUTED PHENYLMETHYL BICYCLOCARBOXYAMIDE COMPOUNDS PFIZER (US) 2011-08-17 EP claimed