SCHEMBL2332522

SCHEMBL2332522

COc1cc([C@@H](C)NC(=O)c2cccc3ccc(C(C)(C)C)nc23)c(Cl)cc1O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.42
MEN1 O00255 6/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
PDE4D Q08499 1/20 0.37
TSHR P16473 1/20 0.37
KDM4E B2RXH2 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
NOD2 Q9HC29 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
KCNMA1 Q12791 1/20 0.36
HIF1A Q16665 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2332116 0.91 MEN1 (0.43) KMT2AMEN1SMN1; SMN2ALDH1A1HPGD
SCHEMBL2329485 0.91 MEN1 (0.43) KMT2AMEN1SMN1; SMN2ALDH1A1HPGD
SCHEMBL2328729 0.88 CYP1A2 (0.39) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL2329497 0.88 CYP1A2 (0.39) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL2330077 0.84 SMN1; SMN2 (0.47) KMT2AMEN1SMN1; SMN2ALDH1A1HPGD
SCHEMBL2332508 0.82 MEN1 (0.41) KMT2AMEN1SMN1; SMN2ALDH1A1HPGD
SCHEMBL2333876 0.80 TRPV1 (0.45) KMT2AHPGDTSHRCYP1A2CYP3A4
SCHEMBL1754350 0.80 TAS1R3 (0.44) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL2330442 0.79 CYP1A2 (0.36) KMT2AMEN1CYP1A2CYP3A4CYP2C19
SCHEMBL2108087 0.74 CYP1A2 (0.38) KMT2AMEN1SMN1; SMN2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222631-B1 SUBSTITUTED PHENYLMETHYL BICYCLOCARBOXYAMIDE COMPOUNDS PFIZER (US) 2011-08-17 EP claimed