SCHEMBL2332508

SCHEMBL2332508

COc1cc(Cl)c([C@@H](C)NC(=O)c2cccc3ccc(C(C)(C)C(F)(F)F)nc23)cc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
PDE4A P27815 2/20 0.35
PDE4B Q07343 2/20 0.35
PDE4C Q08493 2/20 0.35
PDE4D Q08499 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
PDE11A Q9HCR9 1/20 0.35
PDE2A O00408 1/20 0.35
LMNA P02545 2/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
TSHR P16473 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2329485 0.91 MEN1 (0.43) MEN1KMT2ASMN1; SMN2ROCK2ROCK1
SCHEMBL2332116 0.91 MEN1 (0.43) MEN1KMT2ASMN1; SMN2ROCK2ROCK1
SCHEMBL2330442 0.90 CYP1A2 (0.36) MEN1KMT2APDE2APOLBNPC1
SCHEMBL1753951 0.83 TAS1R3 (0.41) MEN1KMT2AROCK2ROCK1TAS1R3
SCHEMBL2332522 0.82 KMT2A (0.42) MEN1KMT2ASMN1; SMN2ROCK2ROCK1
SCHEMBL2329497 0.81 CYP1A2 (0.39) MEN1KMT2AALDH1A1LMNAPOLB
SCHEMBL2328729 0.81 CYP1A2 (0.39) MEN1KMT2AALDH1A1LMNAPOLB
SCHEMBL2326235 0.80 ADORA2A (0.34) PDE2A
SCHEMBL1841391 0.78 CCR1 (0.39) MEN1KMT2AALDH1A1KDM4ERAB9A
SCHEMBL1842345 0.78 ROCK2 (0.35) MEN1KMT2AROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222631-B1 SUBSTITUTED PHENYLMETHYL BICYCLOCARBOXYAMIDE COMPOUNDS PFIZER (US) 2011-08-17 EP claimed