SCHEMBL23315308

SCHEMBL23315308

N#Cc1ccc2c(c1OCc1ccccc1)CCN(C(=O)Cc1ccccc1)C2

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.51
NPC1 O15118 2/20 0.51
ALDH1A1 P00352 3/20 0.47
MEN1 O00255 3/20 0.45
RAB9A P51151 1/20 0.44
S1PR1 P21453 6/20 0.43
PTGDR2 Q9Y5Y4 3/20 0.43
GAA P10253 2/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
HSD17B10 Q99714 1/20 0.42
USP2 O75604 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23315440 0.86 KMT2A (0.51) KMT2ANPC1ALDH1A1MEN1RAB9A
SCHEMBL23315583 0.83 NPC1 (0.62) KMT2ANPC1PTGDR2ALOX15
SCHEMBL23315504 0.78 AGTR2 (0.60)
SCHEMBL23315202 0.78 AGTR2 (0.42) KMT2AALDH1A1MEN1S1PR1GAA
SCHEMBL23315327 0.78 AGTR2 (0.42) KMT2AALDH1A1MEN1S1PR1GAA
SCHEMBL17607347 0.75 ACACB (0.49) KMT2ANPC1
SCHEMBL5132181 0.73 AGTR2 (0.68) KMT2ANPC1MEN1PTGDR2
SCHEMBL11747939 0.72 AGTR2 (0.53) KMT2ANPC1
SCHEMBL29569463 0.71 NPC1 (0.78) KMT2ANPC1ALDH1A1MEN1RAB9A
SCHEMBL25605335 0.71 NPC1 (0.78) KMT2ANPC1ALDH1A1MEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3620454-B1 CARBOXYLIC ACID DERIVATIVE AS AT2R RECEPTOR ANTAGONIST SHANDONG DANHONG PHARMACEUTICAL CO LTD (CN) 2021-05-05 EP disclosed