SCHEMBL23328199

SCHEMBL23328199

Cc1ncc(C)c(C(F)(F)F)n1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
COMT P21964 1/20 0.33
GABBR2 O75899 7/20 0.32
GABBR1 Q9UBS5 7/20 0.32
KDM5B Q9UGL1 1/20 0.32
RAB9A P51151 1/20 0.31
HTT P42858 1/20 0.30
GLP1R P43220 1/20 0.30
SYK P43405 1/20 0.30
PDK2 Q15119 1/20 0.30
AGBL2 Q5U5Z8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ammonia Solution, Strong SCHEMBL29084542 0.98 KDM4E (0.35) KDM4ECOMTGABBR2GABBR1KDM5B
Formamide SCHEMBL21678847 0.89 KDM4E (0.37) KDM4EGABBR2GABBR1KDM5BSYK
SCHEMBL14726084 0.79 NUDT1 (0.32)
SCHEMBL12203584 0.78 NFKB1 (0.44) GLP1R
SCHEMBL6936291 0.78 KDM4E (0.55) KDM4E
SCHEMBL11017429 0.78 KDM4E (0.37) KDM4ECOMTKDM5BHTTAGBL2
SCHEMBL29693635 0.78 KDM4E (0.37) KDM4ECOMTKDM5BHTTAGBL2
SCHEMBL31200389 0.78 MBOAT4 (0.40) KDM4ECOMTGABBR2GABBR1KDM5B
SCHEMBL29693661 0.78 MEN1 (0.35) KDM4ECOMTGABBR2GABBR1KDM5B
SCHEMBL16369420 0.77 AAK1 (0.33) KDM4ECOMTGABBR2GABBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed
US-20230167062-A1 AMIDE COMPOUND CONTAINING SUBSTITUTED ACETOPHENONE STRUCTURAL FRAGMENTS AND PREPARATION METHOD AND APPLICATION THEREOF SHENYANG SINOCHEM AGROCHEMICALS R&D CO., LTD. (CN) 2023-06-01 US disclosed
WO-2023064343-A1 SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF VANQUA BIO, INC. (US) 2023-04-20 WO disclosed
EP-4052576-A1 AMIDE COMPOUND CONTAINING SUBSTITUTED ACETOPHENONE STRUCTURE FRAGMENT, PREPARATION METHOD THEREFOR AND USE THEREOF Shenyang Sinochem Agrochemicals R & D Co., Ltd. (CN) 2022-09-07 EP disclosed
WO-2021082997-A1 AMIDE COMPOUND CONTAINING SUBSTITUTED ACETOPHENONE STRUCTURE FRAGMENT, PREPARATION METHOD THEREFOR AND USE THEREOF 沈阳中化农药化工研发有限公司 2021-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230167062-A1 AMIDE COMPOUND CONTAINING SUBSTITUTED ACETOPHENONE STRUCTURAL FRAGMENTS AND PREPARATION METHOD AND APPLICATION THEREOF AADAC, AAK1, ACLY KDM4E 1998/4885COMT 2654/4885GABBR2 2427/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.