SCHEMBL2333876

SCHEMBL2333876

COc1cc(CNC(=O)c2cccc3ccc(C(C)(C)C)nc23)c(Cl)cc1O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 1/20 0.45
NPC1 O15118 1/20 0.44
HPGD P15428 3/20 0.42
DRD2 P14416 3/20 0.42
DRD4 P21917 3/20 0.42
DRD3 P35462 3/20 0.42
TMEM97 Q5BJF2 3/20 0.42
LMNA P02545 2/20 0.41
KMT2A Q03164 1/20 0.41
TSHR P16473 1/20 0.41
RECQL P46063 1/20 0.41
MAPT P10636 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
PKM P14618 1/20 0.40
CYP2C19 P33261 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2330315 0.90 HPGD (0.44) NPC1HPGDLMNAKMT2ATSHR
SCHEMBL2328736 0.89 TRPV1 (0.45) TRPV1NPC1HPGDDRD2DRD4
SCHEMBL2324504 0.87 MT-CO2 (0.39) TRPV1NPC1HPGDLMNAKMT2A
SCHEMBL2332522 0.80 KMT2A (0.42) NPC1HPGDKMT2ATSHRMAPT
SCHEMBL1754176 0.80 TRPV1 (0.45) TRPV1DRD2DRD3LMNAMAPT
SCHEMBL2333581 0.80 HPGD (0.43) HPGDKMT2A
SCHEMBL2330077 0.73 SMN1; SMN2 (0.47) HPGDLMNAKMT2ATSHR
SCHEMBL1754354 0.72 MAPT (0.43) LMNAMAPT
SCHEMBL2332116 0.72 MEN1 (0.43) NPC1HPGDLMNAKMT2ATSHR
SCHEMBL1753964 0.72 MEN1 (0.49) TRPV1NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2222631-B1 SUBSTITUTED PHENYLMETHYL BICYCLOCARBOXYAMIDE COMPOUNDS PFIZER (US) 2011-08-17 EP claimed