SCHEMBL23364490

SCHEMBL23364490

COc1cc2c(cc1OC)CC(=O)NC2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.56
MAPT P10636 1/20 0.56
GAA P10253 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
KMT2A Q03164 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
EGFR P00533 1/20 0.40
SRC P12931 1/20 0.40
ACHE P22303 1/20 0.40
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30225613 0.89 ACHE (0.49) CYP3A4MAPTGAASMN1; SMN2CRHBP
SCHEMBL23842242 0.89 ACHE (0.49) CYP3A4MAPTGAASMN1; SMN2CRHBP
SCHEMBL10645877 0.82 CYP3A4 (0.62) CYP3A4MAPTGAASMN1; SMN2CRHBP
SCHEMBL24795 0.81 CYP3A4 (0.52) CYP3A4MAPTGAASMN1; SMN2CRHBP
Hydrochloric Acid SCHEMBL30081995 0.80 CYP3A4 (0.50) CYP3A4MAPTGAASMN1; SMN2CRHBP
SCHEMBL13506283 0.77 PDE3B (0.55) GAAPDE3BPDE3ASRCACHE
SCHEMBL6585554 0.74 CYP3A4 (0.71) CYP3A4MAPTGAASMN1; SMN2KMT2A
SCHEMBL30133714 0.74 CHRNB2 (0.37) CYP3A4MAPTGAAPDE3BPDE3A
SCHEMBL24127411 0.74 CHRNB2 (0.37) CYP3A4MAPTGAAPDE3BPDE3A
SCHEMBL4571013 0.73 CYP3A4 (1.00) CYP3A4MAPTGAASMN1; SMN2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021097075-A1 SUBSTITUTED ISOINDOLONYL 2,2'-BIPYRIMIDINYL COMPOUNDS, ANALOGUES THEREOF, AND METHODS USING SAME ARBUTUS BIOPHARMA, INC. (US) 2021-05-20 WO disclosed