SCHEMBL2340709

SCHEMBL2340709

CC#C[C@H](N[C@@H](CSCc1ccccn1)C(=O)NC1(C#N)CC1)C(F)(F)Oc1ccc(SC)cc1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 8/20 0.41
CTSL P07711 8/20 0.40
CTSS P25774 5/20 0.40
CTSB P07858 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15062782 1.00 CTSK (0.41) CTSKCTSLCTSSCTSB
SCHEMBL15062869 0.88 MAPK1 (0.32)
SCHEMBL15062870 0.88 MAPK1 (0.32)
SCHEMBL15062901 0.84 CTSL (0.43) CTSKCTSLCTSSCTSB
SCHEMBL15062902 0.84 CTSL (0.43) CTSKCTSLCTSSCTSB
SCHEMBL15062922 0.78 CTSS (0.45) CTSKCTSLCTSSCTSB
SCHEMBL15062923 0.78 CTSS (0.45) CTSKCTSLCTSSCTSB
SCHEMBL15062865 0.78 MAPK1 (0.36)
SCHEMBL15062866 0.78 MAPK1 (0.36)
SCHEMBL15062929 0.77 CTSL (0.38) CTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2361243-B9 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2014-06-11 EP claimed
EP-2361243-B1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2013-07-03 EP claimed
EP-2361243-B9 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2014-06-11 EP disclosed
EP-2361243-B1 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2013-07-03 EP disclosed
EP-2361243-A2 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS Virobay, Inc. (US) 2011-08-31 EP disclosed
WO-2010056877-A2 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY, INC. (US) 2010-05-20 WO disclosed