SCHEMBL2348397

SCHEMBL2348397

Cc1cccc(C2CC3(CCN(C(=O)Nc4onc(C)c4C)CC3)C2)c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 6/20 0.49
CYP3A4 P08684 5/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP2D6 P10635 1/20 0.43
EDNRA P25101 1/20 0.39
ADAM10 O14672 1/20 0.39
MMP2 P08253 1/20 0.39
MMP9 P14780 1/20 0.39
RAB9A P51151 2/20 0.39
CYP1A2 P05177 5/20 0.39
EPHX2 P34913 1/20 0.38
TSHR P16473 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13355105 0.91 CYP3A4 (0.43) MGLLCYP3A4ALDH1A1CYP2D6CYP1A2
SCHEMBL2341595 0.90 CYP3A4 (0.42) MGLLCYP3A4ALDH1A1CYP2D6EDNRA
SCHEMBL2341768 0.89 MGLL (0.51) MGLLCYP3A4ALDH1A1CYP2D6RAB9A
SCHEMBL2342294 0.89 CYP3A4 (0.41) MGLLCYP3A4ALDH1A1CYP2D6EDNRA
SCHEMBL2345762 0.88 MGLL (0.50) MGLLCYP3A4ALDH1A1CYP2D6CYP1A2
SCHEMBL2341906 0.87 CYP3A4 (0.44) CYP3A4ALDH1A1CYP2D6CYP1A2TSHR
SCHEMBL2346280 0.87 CYP3A4 (0.42) MGLLCYP3A4ALDH1A1CYP2D6RAB9A
SCHEMBL12295576 0.87 MGLL (0.42) MGLLCYP3A4ALDH1A1CYP2D6EDNRA
SCHEMBL2341031 0.86 MGLL (0.52) MGLLCYP3A4ALDH1A1CYP2D6EPHX2
SCHEMBL2347247 0.85 ALDH1A1 (0.41) MGLLCYP3A4ALDH1A1CYP2D6EDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358704-A1 7-azaspiro [3.5]nonane-7-carboxamide compounds as modulators of fatty acid amide hydrolase Pfizer Inc. (US) 2011-08-24 EP claimed
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS PFIZER INC. 2010-05-06 US claimed
WO-2010049841-A1 7-AZASPIRO [3.5] NONANE-7-CARBOXAMIDE COMPOUNDS AS MODULATORS OF FATTY ACID AMIDE HYDROLASE PFIZER INC. (US) 2010-05-06 WO claimed
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS PFIZER INC. 2010-05-06 US disclosed
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS PFIZER INC. 2010-05-06 US disclosed
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS PFIZER INC. 2010-05-06 US disclosed
WO-2010049841-A1 7-AZASPIRO [3.5] NONANE-7-CARBOXAMIDE COMPOUNDS AS MODULATORS OF FATTY ACID AMIDE HYDROLASE PFIZER INC. (US) 2010-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS FAAH, FAAH2, APEH MGLL 298/4885CYP3A4 912/4885ALDH1A1 739/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.