SCHEMBL2348547

SCHEMBL2348547

c1cc2cc(N(c3ccc4sccc4c3)c3ccc4sccc4c3)ccc2s1.c1nc2sccc2s1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.36
CYP2A6 P11509 2/20 0.36
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
CTNNB1 P35222 2/20 0.31
WNT3A P56704 2/20 0.31
KDM1A O60341 1/20 0.31
PTPRC P08575 1/20 0.31
PTPN6 P29350 1/20 0.31
PTPN11 Q06124 1/20 0.31
PTPN22 Q9Y2R2 1/20 0.31
MRGPRX4 Q96LA9 1/20 0.30
CA12 O43570 1/20 0.30
CA2 P00918 1/20 0.30
PER2 O15055 1/20 0.30
CRY1 Q16526 1/20 0.30
CRY2 Q49AN0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL929430 0.82 CYP2A6 (0.48) DYRK1ACYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL219005 0.76
SCHEMBL20386530 0.74 SLC6A2 (0.47) DYRK1ACYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL10051791 0.70 CA2 (0.46) DYRK1ACYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL17010989 0.70 CA2 (0.46) DYRK1ACYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL17740653 0.69 CA2 (0.45) DYRK1ACYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL20408052 0.69 SLC6A2 (0.40) DYRK1ACYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL931734 0.68 ALDH1A1 (0.48) DYRK1A
SCHEMBL10369395 0.68 CYP2A6 (0.46) DYRK1ACYP2A6SLC6A2SLC6A4SLC6A3
SCHEMBL17010919 0.68 CYP2A6 (0.46) DYRK1ACYP2A6SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2361444-A1 MATERIALS Lomox Limited (GB) 2011-08-31 EP disclosed
WO-2009103952-A1 MATERIALS LOMOX LIMITED (GB) 2009-08-27 WO disclosed