SCHEMBL2350355

SCHEMBL2350355

CCOC(=O)CCc1cc(F)c(OCc2cccc(Oc3ccc(OC)cc3)c2)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 13/20 0.52
FFAR4 Q5NUL3 5/20 0.50
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
AKR1C3 P42330 1/20 0.42
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2350121 0.93 FFAR1 (0.53) FFAR1FFAR4THRATHRB
SCHEMBL2354294 0.93 FFAR1 (0.61) FFAR1FFAR4THRATHRB
SCHEMBL2350368 0.93 FFAR1 (0.56) FFAR1FFAR4TDP1THRATHRB
SCHEMBL2350395 0.93 FFAR1 (0.50) FFAR1ALDH1A1MAPTTDP1AKR1C3
SCHEMBL2354216 0.91 FFAR1 (0.51) FFAR1FFAR4THRATHRB
SCHEMBL2354826 0.90 FFAR1 (0.50) FFAR1FFAR4
SCHEMBL2353744 0.89 FFAR1 (0.64) FFAR1FFAR4THRATHRB
SCHEMBL2354053 0.88 FFAR1 (0.56) FFAR1FFAR4ALDH1A1MAPTTDP1
SCHEMBL12394616 0.88 FFAR1 (0.54) FFAR1FFAR4MAPT
SCHEMBL2351981 0.87 PPARG (0.46) FFAR1FFAR4THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8008525-B2 For the 14273 peroxisome proliferator activated receptor; antidiabetic agents, hyperlipidemia, obesity or anorexia; receptor binding assay; drug screening kits TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-08-30 US disclosed
US-20080167378-A1 Receptor Function Regulation Agent TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-07-10 US disclosed
EP-1688138-A1 RECEPTOR FUNCTION REGULATING AGENT Takeda Pharmaceutical Company Limited (JP) 2006-08-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080167378-A1 Receptor Function Regulation Agent GPR119, INSR, GPR88 FFAR1 16/4885FFAR4 17/4885ALDH1A1 3163/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.