SCHEMBL23536110

SCHEMBL23536110

C[Si](C)(C)c1cc(C2CCN(C(=O)O)CC2)no1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD5 Q86SK9 10/20 0.38
SCD O00767 5/20 0.36
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
THRB P10828 1/20 0.34
ALDH1A1 P00352 3/20 0.34
HPGD P15428 3/20 0.34
KDM4E B2RXH2 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 2/20 0.34
TP53 P04637 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CNR2 P34972 1/20 0.33
TSHR P16473 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23536252 0.81 KDM4E (0.51) THRBALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL21080211 0.75 SMYD3 (0.40) NPC1RAB9ASMN1; SMN2TSHR
SCHEMBL21080214 0.75 SMYD3 (0.40) NPC1RAB9ASMN1; SMN2TSHR
SCHEMBL29072056 0.73 SCD5 (0.35) SCD5SCDNPC1RAB9AKDM4E
SCHEMBL2212073 0.71 RAB9A (0.59) SCD5SCDNPC1RAB9AALDH1A1
SCHEMBL21162012 0.67 KDM1A (0.42) NFKB1NFKB2RELA
SCHEMBL3989997 0.67 SCD (0.48) SCD5SCDNPC1RAB9A
SCHEMBL10323271 0.67 KMO (0.45) SCD5ALDH1A1HPGD
SCHEMBL5634920 0.67 EPHX2 (0.57) SMN1; SMN2LMNATSHR
SCHEMBL4706092 0.67 SCD5 (0.34) SCD5SCDNPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021127333-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed
WO-2021127337-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed