SCHEMBL23547459

SCHEMBL23547459

CC(C)Nc1nc(NC2CCN(C(=O)O[C@H]3CCN(C(=O)OC(C)(C)C)C3)CC2)n2ncc(C(C)C)c2n1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 11/20 0.49
CDK7 P50613 6/20 0.49
CDK4 P11802 2/20 0.49
ALDH1A1 P00352 2/20 0.44
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CDK2 P24941 10/20 0.41
PIK3CD O00329 1/20 0.38
ADORA2A P29274 1/20 0.38
CCNH P51946 4/20 0.37
MNAT1 P51948 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23547346 0.94 CDK9 (0.51) CDK9CDK7CDK4ALDH1A1NPC1
SCHEMBL23547464 0.93 ALDH1A1 (0.49) CDK9CDK7CDK4ALDH1A1NPC1
SCHEMBL23547336 0.90 CDK9 (0.52) CDK9CDK7CDK4ALDH1A1NPC1
SCHEMBL23529883 0.90 CDK9 (0.54) CDK9CDK7CDK4ALDH1A1NPC1
SCHEMBL23547379 0.87 CDK9 (0.49) CDK9CDK7CDK4ALDH1A1NPC1
SCHEMBL23547353 0.86 ALDH1A1 (0.51) CDK9CDK7CDK4ALDH1A1NPC1
SCHEMBL31064056 0.84 ALDH1A1 (0.46) CDK9CDK7CDK4ALDH1A1NPC1
SCHEMBL31064050 0.84 ALDH1A1 (0.48) CDK9CDK7CDK4ALDH1A1NPC1
SCHEMBL23547461 0.84 CDK9 (0.45) CDK9CDK7CDK4CDK2
SCHEMBL23547485 0.84 ALDH1A1 (0.52) CDK9CDK7CDK4ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021121390-A1 HETEROCYCLIC COMPOUND, AND PHARMACEUTICAL COMPOSITION THEREOF, PREPARATION METHOD THEREFOR, INTERMEDIATE THEREOF AND APPLICATION THEREOF 苏州信诺维医药科技股份有限公司 2021-06-24 WO disclosed