SCHEMBL2355869

SCHEMBL2355869

Cc1ccc(C(=O)Nc2cc(N3CCCCC3)c(C)c(C(F)(F)F)c2)c(-n2ccnn2)n1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 11/20 0.46
HCRTR2 O43614 10/20 0.46
SCN10A Q9Y5Y9 5/20 0.45
NOTUM Q6P988 2/20 0.44
MALT1 Q9UDY8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2358231 0.90 CHRM1 (0.47) HCRTR1HCRTR2MALT1
SCHEMBL2357713 0.81 HCRTR1 (0.42) HCRTR1HCRTR2MALT1
SCHEMBL2356255 0.80 MALT1 (0.46) MALT1
SCHEMBL2359008 0.80 HCRTR1 (0.41) HCRTR1HCRTR2MALT1
SCHEMBL2363797 0.79 HCRTR1 (0.43) HCRTR1HCRTR2
SCHEMBL2359300 0.78 BRAF (0.45) HCRTR1HCRTR2MALT1
SCHEMBL2356052 0.76 KDM4E (0.45) HCRTR1HCRTR2
SCHEMBL2357650 0.76 CSF1R (0.48) HCRTR1HCRTR2
SCHEMBL2358573 0.74 TRPA1 (0.48) HCRTR1HCRTR2
SCHEMBL2358854 0.72 HCRTR1 (0.38) HCRTR1HCRTR2MALT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350052-A2 ANTIPROLIFERATIVE COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2011-08-03 EP claimed
WO-2010034838-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO claimed