SCHEMBL2358573

SCHEMBL2358573

CCNc1cc(NC(=O)c2ccc(C)nc2-n2ccnn2)cc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 6/20 0.48
HCRTR1 O43613 10/20 0.47
HCRTR2 O43614 10/20 0.46
SORT1 Q99523 1/20 0.44
CYP1A2 P05177 2/20 0.42
JUN P05412 1/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
P2RX1 P51575 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2357713 0.84 HCRTR1 (0.42) HCRTR1HCRTR2SORT1
SCHEMBL2357650 0.81 CSF1R (0.48) HCRTR1HCRTR2
SCHEMBL2357216 0.80 HCRTR1 (0.40) HCRTR1HCRTR2SORT1P2RX1
SCHEMBL2358322 0.79 SORT1 (0.53) HCRTR1HCRTR2SORT1
SCHEMBL2359300 0.76 BRAF (0.45) HCRTR1HCRTR2
SCHEMBL2359008 0.75 HCRTR1 (0.41) HCRTR1HCRTR2SORT1
SCHEMBL2358231 0.75 CHRM1 (0.47) HCRTR1HCRTR2
SCHEMBL2355869 0.74 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL2356052 0.73 KDM4E (0.45) HCRTR1HCRTR2
SCHEMBL2363797 0.72 HCRTR1 (0.43) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350052-A2 ANTIPROLIFERATIVE COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2011-08-03 EP claimed
WO-2010034838-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO claimed