SCHEMBL2359008

SCHEMBL2359008

Cc1ccc(C(=O)Nc2cc(CNC(C)C)c(C)c(C(F)(F)F)c2)c(-n2ccnn2)n1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 14/20 0.41
HCRTR2 O43614 13/20 0.41
MALT1 Q9UDY8 1/20 0.38
SORT1 Q99523 1/20 0.37
TMPRSS4 Q9NRS4 1/20 0.37
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
CMA1 P23946 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2357713 0.82 HCRTR1 (0.42) HCRTR1HCRTR2MALT1SORT1TMPRSS4
SCHEMBL2358854 0.81 HCRTR1 (0.38) HCRTR1HCRTR2MALT1SORT1TMPRSS4
SCHEMBL2355869 0.80 HCRTR1 (0.46) HCRTR1HCRTR2MALT1
SCHEMBL2358231 0.79 CHRM1 (0.47) HCRTR1HCRTR2MALT1
SCHEMBL2363797 0.78 HCRTR1 (0.43) HCRTR1HCRTR2TMPRSS4
SCHEMBL2359300 0.77 BRAF (0.45) HCRTR1HCRTR2MALT1
SCHEMBL2358573 0.75 TRPA1 (0.48) HCRTR1HCRTR2SORT1
SCHEMBL2358322 0.71 SORT1 (0.53) HCRTR1HCRTR2SORT1
SCHEMBL2357650 0.70 CSF1R (0.48) HCRTR1HCRTR2
SCHEMBL2363877 0.69 ALDH1A1 (0.43) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350052-A2 ANTIPROLIFERATIVE COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2011-08-03 EP claimed
WO-2010034838-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO claimed