SCHEMBL2361306

SCHEMBL2361306

COc1cc2[nH]c(-c3c(F)cccc3Cl)nc2cc1-c1nc2cc(C(F)(F)F)ccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 5/20 0.44
PTGES O14684 9/20 0.44
NPBWR1 P48145 2/20 0.43
PTGS1 P23219 1/20 0.42
PDE7A Q13946 1/20 0.42
DGAT1 O75907 1/20 0.40
ORAI1 Q96D31 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2360765 0.81 NPBWR1 (0.48) PTGESNPBWR1PTGS1DGAT1
SCHEMBL2361397 0.80 DGAT1 (0.51) PTGESNPBWR1PTGS1DGAT1
SCHEMBL2342840 0.78 PTGES (0.41) PTGESNPBWR1PTGS1ORAI1
SCHEMBL2361302 0.78 PTGES (0.58) PTGES
SCHEMBL2364623 0.77 USP2 (0.45) PTGES
SCHEMBL2361250 0.77 AMY1A (0.43) AMY1APTGESPDE7ADGAT1ORAI1
SCHEMBL2361260 0.77 PTGES (0.43) PTGESNPBWR1PTGS1
SCHEMBL2361475 0.77 DGAT1 (0.43) AMY1APTGESPTGS1PDE7ADGAT1
SCHEMBL2361234 0.76 PTGES (0.45) AMY1APTGESPDE7ADGAT1ORAI1
SCHEMBL2362184 0.76 AMY1A (0.42) AMY1APTGESPTGS1PDE7ADGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed