SCHEMBL2361981

SCHEMBL2361981

O=Cc1ccc2[nH]c(-c3c(F)cccc3Cl)nc2c1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGES O14684 16/20 0.44
JAK2 O60674 3/20 0.44
CYP2C9 P11712 3/20 0.41
JAK3 P52333 1/20 0.41
CYP2D6 P10635 1/20 0.40
TYK2 P29597 1/20 0.40
PIM1 P11309 1/20 0.40
CSNK2A2 P19784 1/20 0.40
CSNK2B P67870 1/20 0.40
PIM3 Q86V86 1/20 0.40
PIM2 Q9P1W9 1/20 0.40
GUSB P08236 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2361259 0.91 PTGES (0.48) PTGESJAK2CYP2C9CYP2D6TYK2
SCHEMBL2361393 0.81 PTGES (0.47) PTGESJAK2CYP2C9JAK3CYP2D6
SCHEMBL2361320 0.81 PTGES (0.47) PTGESJAK2CYP2C9
SCHEMBL2360992 0.81 PTGES (0.59) PTGESJAK2PIM1CSNK2A2CSNK2B
SCHEMBL2336514 0.80 PTGES (0.45) PTGESJAK2CYP2C9CYP2D6
SCHEMBL2361712 0.80 PTGES (0.50) PTGESJAK2CYP2C9JAK3CYP2D6
SCHEMBL2360771 0.79 PTGES (0.50) PTGESJAK2TYK2
SCHEMBL2362143 0.78 NPBWR1 (0.54)
SCHEMBL2360991 0.78 RHEB (0.52) PTGESJAK2TYK2
SCHEMBL2361888 0.77 AMY1A (0.47) PTGESJAK2CYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed