SCHEMBL2361986

SCHEMBL2361986

O=C(O)[C@H](CC(F)(F)Cc1cccnc1)NCC(F)(F)Oc1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR132 Q9UNW8 8/20 0.42
GAA P10253 1/20 0.39
FDPS P14324 2/20 0.37
SCN9A Q15858 1/20 0.37
KMT2A Q03164 1/20 0.37
ATM Q13315 1/20 0.37
MMP1 P03956 2/20 0.37
MMP9 P14780 2/20 0.37
MMP13 P45452 2/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
CMKLR2 P46091 1/20 0.36
CMKLR1 Q99788 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2361988 1.00 GPR132 (0.42) GPR132GAAFDPSSCN9AKMT2A
SCHEMBL2345194 0.89 FPR2 (0.42) KDM4E
SCHEMBL2345202 0.89 FPR2 (0.42) KDM4E
SCHEMBL2340736 0.86 CASR (0.39)
SCHEMBL2340729 0.86 CASR (0.39)
SCHEMBL2344921 0.85 GPR132 (0.42) GPR132GAASCN9AKMT2AATM
SCHEMBL15062804 0.83 CTSS (0.46)
SCHEMBL15062803 0.83 CTSS (0.46)
SCHEMBL15062860 0.76 ACE (0.42) GPR132KMT2AMMP1MMP9MMP13
SCHEMBL15062928 0.75 CTSK (0.44) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2361243-A2 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS Virobay, Inc. (US) 2011-08-31 EP disclosed
WO-2010056877-A2 HALOALKYL CONTAINING COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY, INC. (US) 2010-05-20 WO disclosed