SCHEMBL23628465

SCHEMBL23628465

NS(=O)(=O)c1ccc(C(=O)N2CC3=C(CN(C(=O)O)C3)C2)cc1F

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.45
CA2 P00918 13/20 0.41
CA1 P00915 12/20 0.41
CA7 P43166 12/20 0.41
CA9 Q16790 12/20 0.41
CA12 O43570 11/20 0.41
CA14 Q9ULX7 11/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TRAP1 Q12931 3/20 0.38
HTT P42858 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
NOD2 Q9HC29 1/20 0.37
ALDH1A1 P00352 1/20 0.36
HSP90B1 P14625 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23628479 0.84 CA12 (0.42) CA2CA1CA7CA9CA12
SCHEMBL21962267 0.82 CA12 (0.55) ENPP2CA2CA1CA7CA9
SCHEMBL23628474 0.80 CA2 (0.39) CA2CA1CA7CA9CA12
SCHEMBL23628467 0.77 CA1 (0.63) CA2CA1CA7CA9CA12
SCHEMBL23628460 0.77 CA2 (0.39) CA2CA1CA7CA9CA12
SCHEMBL23628478 0.75 CA2 (0.41) CA2CA1CA7CA9CA12
SCHEMBL29787231 0.75 NEU3 (0.57) CA2CA1CA7CA9CA12
SCHEMBL2777527 0.75 NEU3 (0.57) CA2CA1CA7CA9CA12
SCHEMBL23628458 0.74 CA2 (0.51) CA2CA1CA7CA9CA12
SCHEMBL23628462 0.74 CA2 (0.58) CA2CA1CA7CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353178-B1 BICYCLIC COMPOUNDS AS DUAL ATX/CA INHIBITORS HOFFMANN LA ROCHE (CH) 2021-07-14 EP claimed