SCHEMBL23628458

SCHEMBL23628458

NS(=O)(=O)c1ccc(S(=O)(=O)N2CC3=C(CN(C(=O)O)C3)C2)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 15/20 0.51
CA1 P00915 8/20 0.40
CA9 Q16790 3/20 0.40
CA7 P43166 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CA12 O43570 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
CA5A P35218 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
USP9X Q93008 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20502523 0.85 ALDH1A1 (0.53) CA2CA1CA9CA7ALDH1A1
SCHEMBL23628462 0.80 CA2 (0.58) CA2CA1CA9CA7CA12
SCHEMBL23628478 0.76 CA2 (0.41) CA2CA1CA9CA7CA12
SCHEMBL21834214 0.76 PKM (0.53) ALDH1A1
SCHEMBL23628465 0.74 ENPP2 (0.45) CA2CA1CA9CA7ALDH1A1
SCHEMBL20502577 0.72 CA2 (0.55) CA2CA1CA9CA7CA12
SCHEMBL30307817 0.71 TGM2 (0.62) CA2ALDH1A1
SCHEMBL23620929 0.71 TGM2 (0.62) CA2ALDH1A1
SCHEMBL23628490 0.71 CA2 (0.49) CA2CA1CA9CA7CA12
SCHEMBL20502276 0.71 CA2 (0.60) CA2CA1CA9CA7CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353178-B1 BICYCLIC COMPOUNDS AS DUAL ATX/CA INHIBITORS HOFFMANN LA ROCHE (CH) 2021-07-14 EP claimed