SCHEMBL23628467

SCHEMBL23628467

NS(=O)(=O)c1ccc(C(=O)N2CC3=C(CN(C(=O)O)C3)C2)cc1

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA1 P00915 20/20 0.63
CA2 P00918 20/20 0.63
CA7 P43166 20/20 0.63
CA9 Q16790 20/20 0.63
CA14 Q9ULX7 19/20 0.63
CA12 O43570 18/20 0.63
CA3 P07451 1/20 0.51
CA6 P23280 1/20 0.51
CYP2C19 P33261 1/20 0.51
CA5A P35218 1/20 0.51
CA5B Q9Y2D0 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17363200 0.80 CA1 (0.61) CA1CA2CA7CA9CA14
SCHEMBL14493373 0.80 CA12 (0.87) CA1CA2CA7CA9CA14
SCHEMBL23628470 0.79 CA2 (0.45) CA1CA2CA7CA9CA14
SCHEMBL23628462 0.77 CA2 (0.58) CA1CA2CA7CA9CA14
SCHEMBL23628479 0.77 CA12 (0.42) CA1CA2CA7CA9CA14
SCHEMBL23628465 0.77 ENPP2 (0.45) CA1CA2CA7CA9CA14
SCHEMBL23628478 0.76 CA2 (0.41) CA1CA2CA7CA9CA14
SCHEMBL18315558 0.76 CA12 (0.60) CA1CA2CA7CA9CA14
SCHEMBL21485402 0.75 CA2 (0.61) CA1CA2CA7CA9CA14
SCHEMBL3570536 0.73 CA12 (0.78) CA1CA2CA7CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353178-B1 BICYCLIC COMPOUNDS AS DUAL ATX/CA INHIBITORS HOFFMANN LA ROCHE (CH) 2021-07-14 EP claimed