SCHEMBL23628478

SCHEMBL23628478

NS(=O)(=O)c1cc(F)c(C(=O)N2CC3=C(CN(C(=O)O)C3)C2)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 18/20 0.41
CA1 P00915 16/20 0.38
CA9 Q16790 12/20 0.38
CA12 O43570 7/20 0.38
CA7 P43166 7/20 0.38
CA14 Q9ULX7 7/20 0.38
CA3 P07451 1/20 0.37
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
HTT P42858 1/20 0.35
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23628462 0.83 CA2 (0.58) CA2CA1CA9CA12CA7
SCHEMBL18668466 0.81 CA2 (0.48) CA2CA1CA9CA12CA7
SCHEMBL23628474 0.76 CA2 (0.39) CA2CA1CA9CA12CA7
SCHEMBL23628458 0.76 CA2 (0.51) CA2CA1CA9CA12CA7
SCHEMBL23628467 0.76 CA1 (0.63) CA2CA1CA9CA12CA7
SCHEMBL23628465 0.75 ENPP2 (0.45) CA2CA1CA9CA12CA7
SCHEMBL20421466 0.73 CA2 (0.50) CA2CA1CA9CA12CA7
SCHEMBL23628490 0.71 CA2 (0.49) CA2CA1CA9CA12CA7
SCHEMBL23628470 0.70 CA2 (0.45) CA2CA1CA9CA12CA7
SCHEMBL23628460 0.70 CA2 (0.39) CA2CA1CA9CA12CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3353178-B1 BICYCLIC COMPOUNDS AS DUAL ATX/CA INHIBITORS HOFFMANN LA ROCHE (CH) 2021-07-14 EP claimed