SCHEMBL2362953

SCHEMBL2362953

O=C(O)CCNC(=O)Cc1ccccc1-c1ccc(Cl)cc1Cl

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.52
GCGR P47871 8/20 0.49
GCG P01275 4/20 0.49
CNR1 P21554 3/20 0.48
SHMT1 P34896 2/20 0.48
SHMT2 P34897 2/20 0.48
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
NPSR1 Q6W5P4 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2364553 0.84 HPGD (0.44) HPGDGCGCNR1NPC1RAB9A
SCHEMBL2363580 0.80 GCGR (0.58) HPGDGCGRGCG
SCHEMBL2363384 0.78 GCGR (0.57) GCGRGCG
SCHEMBL2394244 0.76 CSNK2A2 (0.47) CNR1MEN1KMT2A
SCHEMBL2364901 0.75 GCGR (0.52) HPGDGCGRGCGMEN1KMT2A
SCHEMBL3200958 0.73 AKR1B1 (0.58) HPGDNPSR1
SCHEMBL2804428 0.72 ATM (0.53) HPGD
SCHEMBL29415449 0.72 ATM (0.53) HPGD
SCHEMBL10508515 0.71 CNR1 (0.44) HPGDCNR1MEN1KMT2A
SCHEMBL13602497 0.71 ATM (0.51) HPGDNPC1RAB9ANPSR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349999-A1 ALLOSTERIC PROTEIN KINASE MODULATORS Universität des Saarlandes (DE) 2011-08-03 EP claimed
WO-2010043711-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2010-04-22 WO claimed
WO-2010043711-A1 ALLOSTERIC PROTEIN KINASE MODULATORS UNIVERSITAET DES SAARLANDES (DE) 2010-04-22 WO disclosed