SCHEMBL2363044

SCHEMBL2363044

Cc1cc(C)c(-c2cnccn2)c(C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
PIM1 P11309 1/20 0.40
CYP2A6 P11509 1/20 0.38
LIMK1 P53667 3/20 0.38
LIMK2 P53671 3/20 0.38
TESK1 Q15569 3/20 0.38
TESK2 Q96S53 3/20 0.38
HTT P42858 1/20 0.38
RECQL P46063 1/20 0.38
GAA P10253 1/20 0.37
CCR1 P32246 1/20 0.37
CCR5 P51681 1/20 0.37
CCR8 P51685 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GFER P55789 1/20 0.36
NISCH Q9Y2I1 1/20 0.36
DHODH Q02127 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17755588 0.77 PIM1 (0.45) CYP1A2PIM1CYP2A6HTTRECQL
SCHEMBL8617736 0.77 CYP2D6 (0.43) CYP1A2PIM1CYP2A6HTTRECQL
SCHEMBL28191914 0.72 PIK3R2 (0.44) HTTRECQLGAATDP1NPC1
SCHEMBL3612264 0.72 KDM4E (0.55) CYP1A2HTTCCR1CCR5CCR8
SCHEMBL29633944 0.72 KDM4E (0.55) CYP1A2HTTCCR1CCR5CCR8
SCHEMBL29454745 0.71 NISCH (0.50) CYP1A2PIM1HTTRECQLNPC1
SCHEMBL78566 0.71 NISCH (0.50) CYP1A2PIM1HTTRECQLNPC1
SCHEMBL29598957 0.71 NISCH (0.50) CYP1A2PIM1HTTRECQLNPC1
SCHEMBL18471236 0.71 CYP1A2 (0.44) CYP1A2PIM1CYP2A6HTTRECQL
SCHEMBL26577328 0.70 NOS3 (0.43) GAACCR1CCR5CCR8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1576039-B1 CATALYTIC DEPOLYMERIZATION OF POLYMERS CONTAINING ELECTROPHILIC LINKAGES USING NUCLEOPHILIC REAGENTS IBM (US) 2011-08-03 EP disclosed
US-7544800-B2 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2009-06-09 US disclosed
US-7250510-B2 Transition metal complexes of N-heterocyclic carbenes, method of preparation and use in transition metal catalyzed organic transformations TOTAL SYNTHESIS, LTD. (CA) 2007-07-31 US disclosed
US-7250510-B2 Transition metal complexes of N-heterocyclic carbenes, method of preparation and use in transition metal catalyzed organic transformations TOTAL SYNTHESIS, LTD. (CA) 2007-07-31 US disclosed
US-20070073055-A1 Transition metal complexes of N-heterocyclic carbenes, method of preparation and use in transition metal catalyzed organic transformations TOTAL SYNTHESIS, LTD. (CA) 2007-03-29 US disclosed
US-20070073055-A1 Transition metal complexes of N-heterocyclic carbenes, method of preparation and use in transition metal catalyzed organic transformations TOTAL SYNTHESIS, LTD. (CA) 2007-03-29 US disclosed
US-7053221-B2 Heteroatom-stabilized carbenes and precursors thereto as depolymerization catalysts INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2006-05-30 US disclosed
US-20050288508-A1 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2005-12-29 US disclosed
EP-1576039-A2 CATALYTIC DEPOLYMERIZATION OF POLYMERS CONTAINING ELECTROPHILIC LINKAGES USING NUCLEOPHILIC REAGENTS International Business Machines Corporation (US) 2005-09-21 EP disclosed
US-6916936-B2 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2005-07-12 US disclosed
US-6911546-B2 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2005-06-28 US disclosed
US-20050049418-A1 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents HEDRICK JAMES LUPTON (US) 2005-03-03 US disclosed
WO-2004060987-A2 CATALYTIC DEPOLYMERIZATION OF POLYMERS CONTAINING ELECTROPHILIC LINKAGES USING NUCLEOPHILIC REAGENTS INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2004-07-22 WO disclosed
US-20040127720-A1 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents NATIONAL SCIENCE FOUNDATION 2004-07-01 US disclosed
US-20040127744-A1 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents NATIONAL SCIENCE FOUNDATION 2004-07-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050288508-A1 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents POLL, PNKP, PARN CYP1A2 2496/4885PIM1 1354/4885CYP2A6 4415/4885
US-20050049418-A1 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents POLL, PNKP, PARN CYP1A2 2496/4885PIM1 1354/4885CYP2A6 4415/4885
US-20040127744-A1 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents POLL, PNKP, PARP1 CYP1A2 2467/4885PIM1 1508/4885CYP2A6 4376/4885
US-20040127720-A1 Catalytic depolymerization of polymers containing electrophilic linkages using nucleophilic reagents POLL, PNKP, PARP1 CYP1A2 2467/4885PIM1 1508/4885CYP2A6 4376/4885
US-20070073055-A1 Transition metal complexes of N-heterocyclic carbenes, method of preparation and use in transition metal catalyzed organic transformations NDC1, NBAS, NUDC CYP1A2 102/4885PIM1 1288/4885CYP2A6 726/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.