SCHEMBL23630601

SCHEMBL23630601

CN(C)C(=O)C1CN1S(=O)(=O)c1cccc2cc(N(C)C)ccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 1/20 0.40
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
CNR1 P21554 4/20 0.38
NR1D1 P20393 1/20 0.38
HTR6 P50406 2/20 0.37
CASP3 P42574 1/20 0.34
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
LMNA P02545 1/20 0.33
PRKD3 O94806 1/20 0.33
PRKCG P05129 1/20 0.33
PRKCB P05771 1/20 0.33
PRKCA P17252 1/20 0.33
PRKACA P17612 1/20 0.33
PRKACG P22612 1/20 0.33
PRKACB P22694 1/20 0.33
PRKCH P24723 1/20 0.33
PRKCI P41743 1/20 0.33
PRKCE Q02156 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29948257 1.00 CCR4 (0.40) CCR4HCRTR1HCRTR2CNR1NR1D1
SCHEMBL23630298 0.90 CCR4 (0.41) CCR4HCRTR1HCRTR2CNR1NR1D1
SCHEMBL23630437 0.90 CCR4 (0.41) CCR4HCRTR1HCRTR2CNR1NR1D1
SCHEMBL29948245 0.87 NR1D1 (0.41) CCR4HCRTR1HCRTR2CNR1NR1D1
SCHEMBL30225361 0.87 NR1D1 (0.41) CCR4HCRTR1HCRTR2CNR1NR1D1
SCHEMBL29948239 0.87 NR1D1 (0.41) CCR4HCRTR1HCRTR2CNR1NR1D1
SCHEMBL23630431 0.87 NR1D1 (0.41) CCR4HCRTR1HCRTR2CNR1NR1D1
SCHEMBL23630459 0.79 KMT2A (0.55)
SCHEMBL29948271 0.79 KMT2A (0.55)
SCHEMBL23630364 0.77 CASP3 (0.43) CCR4CASP3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021141506-A1 AROMATIC SULPHONAMIDES DERIVATIVES THAT INHIBITS PDI A1, THEIR SYNTHESIS AND USE Uniwersytet Jagielloński (PL) 2021-07-15 WO claimed
WO-2021141506-A1 AROMATIC SULPHONAMIDES DERIVATIVES THAT INHIBITS PDI A1, THEIR SYNTHESIS AND USE Uniwersytet Jagielloński (PL) 2021-07-15 WO disclosed