SCHEMBL2363877

SCHEMBL2363877

Cc1ccc(C(=O)Nc2cnn(C(C)C)c2)c(-n2ccnn2)n1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
HTT P42858 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
HCRTR1 O43613 11/20 0.43
HCRTR2 O43614 10/20 0.43
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
NAMPT P43490 1/20 0.40
RPS6KA2 Q15349 1/20 0.39
FPR2 P25090 1/20 0.39
MAPK8 P45983 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37
MAPK14 Q16539 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28046546 0.74 HCRTR1 (0.56) HCRTR1HCRTR2
SCHEMBL1586336 0.73 HCRTR1 (0.55) HCRTR1HCRTR2
SCHEMBL2355558 0.72 HCRTR1 (0.54) HCRTR1HCRTR2
SCHEMBL2359008 0.69 HCRTR1 (0.41) HCRTR1HCRTR2
SCHEMBL2358573 0.69 TRPA1 (0.48) HCRTR1HCRTR2
SCHEMBL2359300 0.69 BRAF (0.45) HCRTR1HCRTR2LMNAMAPT
SCHEMBL2358684 0.69 NPC1 (0.52) ALDH1A1HTTNPC1RAB9AHCRTR1
SCHEMBL2358322 0.68 SORT1 (0.53) HCRTR1HCRTR2
SCHEMBL2357713 0.68 HCRTR1 (0.42) HCRTR1HCRTR2
SCHEMBL4285419 0.67 NPC1 (0.69) ALDH1A1HTTNPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2350052-A2 ANTIPROLIFERATIVE COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2011-08-03 EP claimed
WO-2010034838-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO claimed