SCHEMBL2364222

SCHEMBL2364222

CCOC=C(C(C)=O)C(=O)OCC.CSC(=N)N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLO1 Q04760 2/20 0.50
NPSR1 Q6W5P4 5/20 0.39
ALDH1A1 P00352 6/20 0.35
GAA P10253 1/20 0.35
CYP2D6 P10635 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 9/20 0.34
KMT2A Q03164 9/20 0.34
MAPK1 P28482 2/20 0.33
ALOX15 P16050 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
MAPT P10636 7/20 0.33
KDM4E B2RXH2 3/20 0.33
HSP90AA1 P07900 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 2/20 0.32
BLM P54132 1/20 0.32
USP2 O75604 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1186672 0.85 GLO1 (0.67) GLO1NPSR1ALDH1A1GAACYP2D6
SCHEMBL1186674 0.85 GLO1 (0.67) GLO1NPSR1ALDH1A1GAACYP2D6
SCHEMBL4197379 0.85 GLO1 (0.67) GLO1NPSR1ALDH1A1GAACYP2D6
SCHEMBL11101309 0.77 NPSR1 (0.48) GLO1NPSR1ALDH1A1GAACYP2D6
SCHEMBL14827720 0.77 NPSR1 (0.48) GLO1NPSR1ALDH1A1GAACYP2D6
SCHEMBL50838 0.76 NPSR1 (0.56) GLO1NPSR1ALDH1A1GAACYP2D6
SCHEMBL24937270 0.75 GLO1 (0.57) GLO1NPSR1ALDH1A1GAACYP2D6
SCHEMBL28786257 0.75 GLO1 (0.57) GLO1NPSR1ALDH1A1GAACYP2D6
SCHEMBL29636860 0.75 GLO1 (0.53) GLO1NPSR1ALDH1A1GAACYP2D6
SCHEMBL11651951 0.74 GLO1 (0.50) GLO1NPSR1ALDH1A1GAACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2352732-A1 2, 5-DIAMINO-SUBSTITUTED PYRIDO Ý4, 3-D¨PYRIMIDINES AS AUTOTAXIN INHIBITORS AGAINST CANCER Merck Patent GmbH (DE) 2011-08-10 EP disclosed