SCHEMBL2364703

SCHEMBL2364703

Cc1ccc(-c2c[nH]c(-c3ccc4[nH]c(-c5c(F)cccc5Cl)nc4c3)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGES O14684 15/20 0.48
CYP2C9 P11712 3/20 0.43
CYP2D6 P10635 1/20 0.43
JAK2 O60674 1/20 0.38
PTGS1 P23219 1/20 0.36
DGAT1 O75907 1/20 0.36
MAPK14 Q16539 2/20 0.36
DHODH Q02127 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2361234 0.84 PTGES (0.45) PTGESCYP2C9CYP2D6DGAT1
SCHEMBL14146990 0.83 PTGES (0.42) PTGESCYP2C9DGAT1
SCHEMBL12446417 0.83 NPBWR1 (0.46) PTGESPTGS1DGAT1
SCHEMBL2361014 0.77 PTGES (0.43) PTGESCYP2C9CYP2D6JAK2DGAT1
SCHEMBL2361475 0.77 DGAT1 (0.43) PTGESCYP2C9CYP2D6PTGS1DGAT1
SCHEMBL3796104 0.77 PTGES (0.48) PTGESJAK2
SCHEMBL2361250 0.76 AMY1A (0.43) PTGESCYP2C9CYP2D6JAK2DGAT1
SCHEMBL2360765 0.75 NPBWR1 (0.48) PTGESPTGS1DGAT1
SCHEMBL2361558 0.75 PTGES (0.53) PTGESCYP2C9CYP2D6JAK2DGAT1
SCHEMBL29662800 0.75 PTGES (0.43) PTGESCYP2C9JAK2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed