SCHEMBL2365575

SCHEMBL2365575

CCCN(C(=O)O)c1cccc(Cc2nn(-c3ccn(C)n3)ccc2=O)c1

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.32
KDM5A P29375 1/20 0.31
KDM2B Q8NHM5 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
ALDH1A1 P00352 3/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
PAX8 Q06710 2/20 0.31
JAK2 O60674 1/20 0.31
HTT P42858 1/20 0.31
PARP1 P09874 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
GRM2 Q14416 1/20 0.31
GPX4 P36969 1/20 0.30
JMJD6 Q6NYC1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13274570 0.92 TP53 (0.36) TP53KDM5AKDM2BKDM4CKDM5B
SCHEMBL2220897 0.88 KDM5A (0.33) KDM5AKDM2BKDM4CKDM5BALDH1A1
SCHEMBL2221099 0.85 TP53 (0.38) TP53ALDH1A1NPC1RAB9APAX8
SCHEMBL2221804 0.84 ENPP2 (0.35) TP53ALDH1A1NPC1RAB9APAX8
SCHEMBL2223717 0.83 KMT2A (0.33) TP53ALDH1A1NPC1RAB9APAX8
SCHEMBL2221341 0.83 PDE10A (0.33) TP53ALDH1A1NPC1RAB9APAX8
SCHEMBL2223741 0.82 PDE10A (0.34) TP53ALDH1A1NPC1RAB9APAX8
SCHEMBL2219994 0.82 MEN1 (0.37) ALDH1A1HTTPTGDR2
SCHEMBL2222006 0.82 GRM2 (0.40) TP53HTTGRM2
SCHEMBL2220317 0.80 GRM5 (0.38) GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011084402-A1 TYROSINE KINASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-07-14 WO disclosed