SCHEMBL2367200

SCHEMBL2367200

Cc1ccc(C)c2c1[nH]c1c(NS(=O)(=O)c3cccc(C(F)(F)F)c3)cccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.53
HSD17B2 P37059 1/20 0.52
LMNA P02545 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
MEN1 O00255 1/20 0.50
GAA P10253 1/20 0.50
KMT2A Q03164 1/20 0.50
SLC40A1 Q9NP59 1/20 0.48
PTGES2 Q9H7Z7 2/20 0.47
ACLY P53396 1/20 0.46
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
MMP1 P03956 1/20 0.45
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
MMP8 P22894 1/20 0.45
MMP13 P45452 1/20 0.45
CKS1B P61024 2/20 0.45
SKP2 Q13309 2/20 0.45
CCR2 P41597 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2367599 0.84 RECQL (0.51) LMNAMEN1GAAKMT2ASLC40A1
SCHEMBL2406982 0.82 HSD17B2 (0.44) CLK1HSD17B2LMNANPSR1CA1
SCHEMBL2368002 0.81 MEN1 (0.58) CLK1LMNANPSR1MEN1GAA
SCHEMBL2367251 0.80 KEAP1 (0.54) LMNANPSR1MEN1KMT2ASLC40A1
SCHEMBL26844377 0.80 CRBN (0.56) CLK1HSD17B2LMNANPSR1MEN1
SCHEMBL2367596 0.78 CA1 (0.56) LMNACA1CA2CRBN
SCHEMBL2367468 0.78 HTR6 (0.49) LMNAMEN1KMT2ACA1CA2
SCHEMBL2367619 0.78 ALDH1A1 (0.56) LMNAGAASLC40A1CA1CA2
SCHEMBL2367180 0.78 HSD17B2 (0.39) HSD17B2LMNANPSR1GAACA1
SCHEMBL2367618 0.76 KEAP1 (0.57) LMNANPSR1GAAKMT2ASLC40A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2366687-B1 Benzenesulfonamide derivatives and pharmaceutical composition thereof PURZER PHARMACEUTICAL CO LTD (CN) 2015-11-04 EP disclosed
EP-2366687-B1 Benzenesulfonamide derivatives and pharmaceutical composition thereof PURZER PHARMACEUTICAL CO LTD (CN) 2015-11-04 EP disclosed
US-8173693-B2 Benzenesulfonamide derivatives and pharmaceutical composition thereof PURZER PHARMACEUTICAL CO., LTD. (TW) 2012-05-08 US disclosed
US-8173693-B2 Benzenesulfonamide derivatives and pharmaceutical composition thereof PURZER PHARMACEUTICAL CO., LTD. (TW) 2012-05-08 US disclosed
US-8173693-B2 Benzenesulfonamide derivatives and pharmaceutical composition thereof PURZER PHARMACEUTICAL CO., LTD. (TW) 2012-05-08 US disclosed
CN-102199148-A Benzenesulfonamide derivatives and pharmaceutical compositions thereof PURZER PHARMACEUTICAL CO LTD 2011-09-28 CN disclosed
US-20110230651-A1 Benzenesulfonamide derivatives and pharmaceutical composition therof PURZER PHARMACEUTICAL CO., LTD. (TW) 2011-09-22 US disclosed
US-20110230651-A1 Benzenesulfonamide derivatives and pharmaceutical composition therof PURZER PHARMACEUTICAL CO., LTD. (TW) 2011-09-22 US disclosed
US-20110230651-A1 Benzenesulfonamide derivatives and pharmaceutical composition therof PURZER PHARMACEUTICAL CO., LTD. (TW) 2011-09-22 US disclosed
EP-2366687-A2 Benzenesulfonamide derivatives and pharmaceutical composition thereof Purzer Pharmaceutical Co., Ltd. (CN) 2011-09-21 EP disclosed
EP-2366687-A2 Benzenesulfonamide derivatives and pharmaceutical composition thereof Purzer Pharmaceutical Co., Ltd. (CN) 2011-09-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110230651-A1 Benzenesulfonamide derivatives and pharmaceutical composition therof CCNI, CCNE1, CCND1 CLK1 4251/4885HSD17B2 3109/4885LMNA 1894/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.