SCHEMBL2369264

SCHEMBL2369264

CCc1sc2ncncc2c1-c1ccoc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.37
TMIGD3 P0DMS9 1/20 0.37
CYP1A2 P05177 14/20 0.36
CYP3A4 P08684 14/20 0.36
CYP2C19 P33261 12/20 0.36
CYP2D6 P10635 10/20 0.36
MEN1 O00255 7/20 0.36
KMT2A Q03164 7/20 0.36
ALOX15 P16050 5/20 0.36
ALDH1A1 P00352 11/20 0.36
CLK4 Q9HAZ1 10/20 0.36
USP2 O75604 5/20 0.36
CYP2C9 P11712 5/20 0.36
HSD17B10 Q99714 7/20 0.36
TSHR P16473 5/20 0.36
LMNA P02545 3/20 0.36
GLA P06280 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6358968 0.75 ADORA1 (0.34) ADORA1TMIGD3ADORA2A
SCHEMBL2369044 0.68 MCL1 (0.34) ADORA1TMIGD3CYP1A2CYP3A4CYP2C19
SCHEMBL3384503 0.68 MCL1 (0.36) CYP2C19MEN1KMT2AALOX15ALDH1A1
SCHEMBL3384508 0.67 SMN1; SMN2 (0.58) CYP1A2CYP3A4CYP2C19CYP2D6MEN1
SCHEMBL2368933 0.61 MAPK1 (0.44) MEN1KMT2AALDH1A1TSHRKDM4E
SCHEMBL27386212 0.60 SELE (0.36) CYP1A2ALDH1A1CYP2C9TSHRLMNA
SCHEMBL29619599 0.59 CYP1A2 (0.42) CYP1A2CYP3A4CYP2C19CYP2D6MEN1
SCHEMBL2369352 0.58 ATM (0.37) MEN1KMT2AALDH1A1USP2HSD17B10
SCHEMBL2056343 0.58 CYP1A2 (0.39) ADORA1CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL2716516 0.57 CYP11B1 (0.59) ADORA1CYP1A2CYP3A4CYP2D6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8022076-B2 Thieno[2,3-d]pyrimidine derivatives as potassium channel modulators; antiarrhythmia agents XENTION LIMITED (GB) 2011-09-20 US disclosed