SCHEMBL2369924

SCHEMBL2369924

O=C(O)N(c1ccccc1)c1ccc(-c2ccnc(N3CC4CCC(C3)O4)n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 1/20 0.48
HCRTR1 O43613 16/20 0.47
HCRTR2 O43614 16/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14471461 0.79 HCRTR1 (0.45) HCRTR1HCRTR2
SCHEMBL15144965 0.77 PORCN (0.44) HCRTR1HCRTR2
SCHEMBL2370406 0.77 MTOR (0.46) HCRTR1HCRTR2
SCHEMBL2369667 0.74 MTOR (0.55)
SCHEMBL8533161 0.74 AGTR2 (0.43) AGTR2HCRTR1HCRTR2
SCHEMBL2369920 0.73 MTOR (0.48)
SCHEMBL2369911 0.73 MTOR (0.48)
SCHEMBL2370567 0.72 MTOR (0.56)
SCHEMBL2369988 0.71 MTOR (0.56)
SCHEMBL22917166 0.70 AGTR2 (0.70) AGTR2HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9249129-B2 Morpholino substituted urea derivatives as mTOR inhibitors CELLZOME LIMITED (GB) 2016-02-02 US disclosed
US-20130196982-A1 MORPHOLINO SUBSTITUTED UREA DERIVATIVES AS MTOR INHIBITORS CELLZOME LIMITED (GB) 2013-08-01 US disclosed
WO-2011107585-A1 MORPHOLINO SUBSTITUTED UREA DERIVATIVES AS MTOR INHIBITORS CELLZOME LIMITED (GB) 2011-09-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130196982-A1 MORPHOLINO SUBSTITUTED UREA DERIVATIVES AS MTOR INHIBITORS MTOR, EIF4E, EIF4A1 AGTR2 3149/4885HCRTR1 3325/4885HCRTR2 3843/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.