SCHEMBL2370366

SCHEMBL2370366

COc1cccc(CCC2(N)CCCC2)c1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.57
HRH3 Q9Y5N1 3/20 0.52
SIGMAR1 Q99720 1/20 0.51
AOC3 Q16853 1/20 0.51
CHRM2 P08172 2/20 0.50
CHRM1 P11229 2/20 0.50
CHRM3 P20309 2/20 0.50
IDO1 P14902 2/20 0.49
AGXT P21549 2/20 0.49
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2371058 0.81 TAAR1 (0.52) TAAR1HRH3SIGMAR1AOC3IDO1
SCHEMBL1820761 0.80 TSHR (0.50) TAAR1HRH3SIGMAR1AOC3IDO1
Hydrochloric Acid SCHEMBL3964945 0.78 TSHR (0.49) TAAR1HRH3SIGMAR1AOC3IDO1
SCHEMBL3163183 0.78 TAAR1 (0.54) TAAR1HRH3SIGMAR1AOC3CHRM2
SCHEMBL723511 0.76 TAAR1 (0.77) TAAR1HRH3SIGMAR1AOC3CHRM2
SCHEMBL30080050 0.76 TAAR1 (0.77) TAAR1HRH3SIGMAR1AOC3CHRM2
SCHEMBL21058245 0.75 MAOA (0.52) TAAR1
SCHEMBL29966158 0.74 MTNR1A (0.48) TAAR1HRH3SIGMAR1AOC3CHRM2
SCHEMBL29092222 0.74 MTNR1A (0.48) TAAR1HRH3SIGMAR1AOC3CHRM2
SCHEMBL1824117 0.74 TAAR1 (0.55) TAAR1HRH3SIGMAR1AOC3IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011116356-A2 POSITIVE ALLOSTERIC MODULATORS OF GROUP II MGLURS SANFORD-BURNHAM MEDICAL RESEARCH INSTITUTE (US) 2011-09-22 WO disclosed