SCHEMBL23715809

SCHEMBL23715809

NC(=O)C(Nc1ccc(Cl)c(Cl)c1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
MMP8 P22894 1/20 0.47
MMP14 P50281 1/20 0.47
CA14 Q9ULX7 1/20 0.47
EPHX1 P07099 1/20 0.46
EPHX2 P34913 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
PDGFRA P16234 1/20 0.46
MAPK1 P28482 1/20 0.46
MAPKAPK2 P49137 1/20 0.46
RPS6KA1 Q15418 1/20 0.46
AURKB Q96GD4 1/20 0.46
CSNK1G1 Q9HCP0 1/20 0.46
MAPK14 Q16539 1/20 0.46
GAA P10253 1/20 0.44
S1PR3 Q99500 6/20 0.44
S1PR4 O95977 3/20 0.44
S1PR2 O95136 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7584703 0.87 NPC1 (0.53) NPC1RAB9AMMP8MMP14CA14
SCHEMBL17664140 0.83 RAB9A (0.56) NPC1RAB9AMMP8MMP14CA14
SCHEMBL16838610 0.83 MAPT (0.50) NPC1RAB9AEPHX1CYP3A4CYP2C9
SCHEMBL17663794 0.82 NPC1 (0.51) NPC1RAB9AEPHX1EPHX2GAA
SCHEMBL2537569 0.81 CYP3A4 (0.54) EPHX1CYP3A4CYP2C9PDGFRAMAPK1
SCHEMBL23716088 0.80 ALDH1A1 (0.47) NPC1RAB9ACYP3A4CYP2C9PDGFRA
SCHEMBL17663823 0.80 MEN1 (0.55) NPC1RAB9AEPHX1EPHX2GAA
SCHEMBL11260997 0.78 CYP3A4 (0.48) EPHX1CYP3A4CYP2C9PDGFRAMAPK1
SCHEMBL23716261 0.77 MEN1 (0.49) NPC1RAB9AMMP8MMP14CA14
SCHEMBL17664138 0.77 ALDH1A1 (0.56) NPC1RAB9AMMP8MMP14CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209732-B1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS SCRIPPS RESEARCH INST (US) 2021-08-04 EP disclosed