SCHEMBL23716252

SCHEMBL23716252

Cc1cnc(Cc2ccc(Cl)c(F)c2)c(F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 1/20 0.35
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
P2RX7 Q99572 1/20 0.34
PARP1 P09874 1/20 0.33
KCNH2 Q12809 1/20 0.33
FPR2 P25090 2/20 0.33
PROKR1 Q8TCW9 2/20 0.33
HCRTR2 O43614 1/20 0.33
ANO1 Q5XXA6 1/20 0.33
GRM2 Q14416 1/20 0.33
AKT1 P31749 1/20 0.32
QPCT Q16769 2/20 0.32
QPCTL Q9NXS2 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
ALOX5AP P20292 1/20 0.32
GPR52 Q9Y2T5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17664039 0.90 RAPGEF4 (0.40) RAPGEF4CYP11B1CYP11B2P2RX7PARP1
SCHEMBL17664085 0.84 PARP1 (0.37) PARP1GRM2QPCTQPCTLMAPT
SCHEMBL17664049 0.81 PARP1 (0.35) RAPGEF4P2RX7PARP1KCNH2FPR2
SCHEMBL23715992 0.79 RAPGEF4 (0.33) RAPGEF4P2RX7PARP1KCNH2FPR2
SCHEMBL17664040 0.79 NPC1 (0.37) RAPGEF4KCNH2HCRTR2NPC1RAB9A
SCHEMBL17664035 0.78 S1PR1 (0.38) RAPGEF4P2RX7PARP1KCNH2FPR2
SCHEMBL23715848 0.75 RAB9A (0.38) RAB9AMAPTMAPK1
SCHEMBL17664392 0.72 PARP1 (0.45) P2RX7PARP1ANO1GRM2NPC1
SCHEMBL29636159 0.71 CCR1 (0.34) ALOX5AP
SCHEMBL16039165 0.71 CCR1 (0.34) ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209732-B1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS SCRIPPS RESEARCH INST (US) 2021-08-04 EP disclosed