SCHEMBL23716678

SCHEMBL23716678

Cc1cccc(C)c1C(=O)N1CC[C@H](Oc2cccc(N)c2)C1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SPR P35270 2/20 0.48
CCR5 P51681 4/20 0.47
EPHX2 P34913 1/20 0.41
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
CHRM3 P20309 2/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
PIK3CD O00329 2/20 0.40
PIK3CA P42336 2/20 0.40
PDE2A O00408 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
OPRK1 P41145 2/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
OPRM1 P35372 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23734784 0.88 ALDH1A1 (0.51) SPREPHX2KMT2A
SCHEMBL23734850 0.86 SMN1; SMN2 (0.48) SPREPHX2HCRTR1HCRTR2KMT2A
SCHEMBL23734774 0.85 SPR (0.46) SPRCCR5OPRK1KCNH2
SCHEMBL22735458 0.84 HCRTR1 (0.48) SPREPHX2HCRTR1HCRTR2KMT2A
SCHEMBL22735588 0.84 HTT (0.51) EPHX2KMT2AMEN1HRH3OPRK1
SCHEMBL23734969 0.84 HTT (0.51) EPHX2KMT2AMEN1HRH3OPRK1
SCHEMBL22771999 0.83 SLC6A2 (0.48) SPRCCR5KMT2A
SCHEMBL596167 0.82 OPRK1 (0.44) SPREPHX2CHRM3KMT2AMEN1
SCHEMBL596166 0.82 OPRK1 (0.44) SPREPHX2CHRM3KMT2AMEN1
SCHEMBL23734990 0.80 HCRTR1 (0.42) CCR5HCRTR1HCRTR2KMT2AOPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3594202-B1 SUBSTITUTED PYRROLIDINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2021-08-11 EP disclosed
EP-3594202-B1 SUBSTITUTED PYRROLIDINE COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2021-08-11 EP disclosed