SCHEMBL23718330

SCHEMBL23718330

Cn1cnc2nnn(C)c2c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 11/20 0.41
ADORA2A P29274 2/20 0.38
ADORA2B P29275 2/20 0.38
GDA Q9Y2T3 2/20 0.38
PIK3CD O00329 1/20 0.38
POLB P06746 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CNR1 P21554 1/20 0.38
ACHE P22303 1/20 0.38
ADORA1 P30542 1/20 0.38
NTSR1 P30989 1/20 0.38
MC3R P41968 1/20 0.38
NOTUM Q6P988 1/20 0.38
SIRT3 Q9NTG7 1/20 0.38
NR2E1 Q9Y466 1/20 0.38
CYP3A4 P08684 2/20 0.36
BLM P54132 2/20 0.36
PMP22 Q01453 2/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20203371 0.79 TRPA1 (0.39) TRPA1
SCHEMBL20203174 0.77 ADORA2A (0.48) TRPA1ADORA2AADORA2BGDAPIK3CD
SCHEMBL25165827 0.74 TRPA1 (0.36) TRPA1
Hydrochloric Acid SCHEMBL18704207 0.73 ADORA2B (0.48) TRPA1ADORA2BPOLBLMNA
SCHEMBL17164066 0.68 ALDH1A1 (0.45) ADORA2APOLBBLMALDH1A1LMNA
SCHEMBL25165828 0.68 ADORA2A (0.50) TRPA1ADORA2AADORA2BGDAPIK3CD
SCHEMBL20203177 0.68 PIK3CD (0.37) ADORA2AADORA2BGDAPIK3CDPOLB
SCHEMBL9604644 0.63 ADORA2A (0.46) ADORA2AADORA2BADORA1LMNA
SCHEMBL14930043 0.61 ADORA2A (0.40) ADORA2AADORA2BGDAPIK3CDPOLB
SCHEMBL10328327 0.61 ACVR1 (0.51) TRPA1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3544979-B1 OXADIAZOLONES AS TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS HOFFMANN LA ROCHE (CH) 2021-08-04 EP disclosed