SCHEMBL23729095

SCHEMBL23729095

C/C=C(\C)Nc1cc2cccnc2cc1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
PDGFRB P09619 1/20 0.41
PDGFRA P16234 1/20 0.41
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
NPC1 O15118 4/20 0.40
POLB P06746 3/20 0.40
MAPT P10636 1/20 0.40
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
RAB9A P51151 2/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
PRKDC P78527 1/20 0.39
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
PLK1 P53350 1/20 0.38
NOTUM Q6P988 2/20 0.38
KDM4E B2RXH2 1/20 0.37
BRAF P15056 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8404544 0.73 ALDH1A1 (0.61) ALDH1A1PDGFRBPDGFRAMEN1KMT2A
SCHEMBL31186675 0.73 ALDH1A1 (0.61) ALDH1A1PDGFRBPDGFRAMEN1KMT2A
SCHEMBL246244 0.71 ALDH1A1 (0.53) ALDH1A1PDGFRBPDGFRAMEN1KMT2A
SCHEMBL12047115 0.71 SLC40A1 (0.51) MEN1KMT2ANPC1POLBMAPT
SCHEMBL20278424 0.70 ALDH1A1 (0.49) ALDH1A1PDGFRBPDGFRAMEN1KMT2A
SCHEMBL26235009 0.69 ALDH1A1 (0.47) ALDH1A1PDGFRBPDGFRAMEN1KMT2A
SCHEMBL29870301 0.69 NPC1 (0.49) ALDH1A1PDGFRBPDGFRAMEN1KMT2A
SCHEMBL5545370 0.67 ALDH1A1 (0.53) ALDH1A1PDGFRBPDGFRAMEN1KMT2A
SCHEMBL5542743 0.67 ALDH1A1 (0.53) ALDH1A1PDGFRBPDGFRAMEN1KMT2A
SCHEMBL3344562 0.67 CASP6 (0.62) ALDH1A1PDGFRBPDGFRAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3205650-B1 EGFR INHIBITOR, AND PREPARATION AND APPLICATION THEREOF SHANGHAI HANSOH BIOMEDICAL CO LTD (CN) 2021-08-04 EP disclosed