SCHEMBL23742604

SCHEMBL23742604

Fc1ccccc1Nc1nc(-c2cccc(-c3nnn[nH]3)c2)cs1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 1/20 0.46
CTRB1 P17538 1/20 0.43
CTRC Q99895 1/20 0.43
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
POLB P06746 2/20 0.43
NSD2 O96028 1/20 0.43
ALPL P05186 1/20 0.43
ALPI P09923 1/20 0.43
CASP6 P55212 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
OPRM1 P35372 1/20 0.43
KIT P10721 2/20 0.42
PLAU P00749 1/20 0.41
CYP1A1 P04798 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP1B1 Q16678 1/20 0.41
ROCK1 Q13464 1/20 0.41
CSNK2A1 P68400 1/20 0.41
RAB9A P51151 5/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23742582 0.80 CYP1A1 (0.57) CCR4CTRB1CTRCMEN1KMT2A
SCHEMBL25959089 0.79 CCR4 (0.54) CCR4CTRB1CTRCMEN1KMT2A
SCHEMBL23742583 0.78 CCR4 (0.67) CCR4MEN1KMT2ACYP1A1CYP1A2
SCHEMBL23742661 0.78 MAPT (0.58) CCR4CTRB1CTRCMEN1KMT2A
SCHEMBL23742615 0.78 VCP (0.64) CCR4CTRB1CTRCMEN1KMT2A
SCHEMBL23742660 0.77 RAB9A (0.47) CCR4CTRB1CTRCMEN1KMT2A
SCHEMBL23742607 0.77 CTRB1 (0.52) CCR4CTRB1CTRCMEN1KMT2A
SCHEMBL23742674 0.76 MEN1 (0.57) CCR4CTRB1CTRCMEN1KMT2A
SCHEMBL23742622 0.76 CFTR (0.59) CCR4CTRB1CTRCMEN1KMT2A
SCHEMBL23742648 0.75 CCR4 (0.50) CCR4CTRB1CTRCMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230286933-A1 2,5-ARYL-THIAZOLE ANALOGS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES SOUTHERN RES INST (US) 2023-09-14 US disclosed
US-11718593-B2 2,5-aryl-thiazole analogs for the treatment of neurodegenerative diseases SOUTHERN RESEARCH INSTITUTE (US) 2023-08-08 US disclosed
US-20210246110-A1 2,5-ARYL-THIAZOLE ANALOGS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES SOUTHERN RESEARCH INSTITUTE 2021-08-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11718593-B2 2,5-aryl-thiazole analogs for the treatment of neurodegenerative diseases SMN1; SMN2, TDP2, TDP1 CCR4 4072/4885CTRB1 2158/4885CTRC 4016/4885
US-20210246110-A1 2,5-ARYL-THIAZOLE ANALOGS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES SMN1; SMN2, TDP2, TDP1 CCR4 4072/4885CTRB1 2158/4885CTRC 4016/4885
US-20230286933-A1 2,5-ARYL-THIAZOLE ANALOGS FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES SMN1; SMN2, TDP2, TDP1 CCR4 4072/4885CTRB1 2158/4885CTRC 4016/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.