SCHEMBL2376172

SCHEMBL2376172

COc1ccc(CNC(C)C(=O)O)cc1O

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.58
ALOX15 P16050 2/20 0.58
KDM4E B2RXH2 2/20 0.58
CYP3A4 P08684 2/20 0.58
TSHR P16473 2/20 0.58
RAB9A P51151 1/20 0.58
TRPV1 Q8NER1 4/20 0.56
ALOX12 P18054 1/20 0.55
ALDH1A1 P00352 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
TUBB1 Q9H4B7 1/20 0.49
MAPK1 P28482 1/20 0.48
CYP1A2 P05177 1/20 0.48
NFKB1 P19838 1/20 0.48
CD274 Q9NZQ7 2/20 0.47
LDHA P00338 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27471328 0.84 CD274 (0.57) GAAKDM4ETSHRALDH1A1TDP1
SCHEMBL9462879 0.83 ERCC1 (0.59) GAAALOX15KDM4ECYP3A4TSHR
SCHEMBL3721209 0.79 TRPV1 (0.69) GAAALOX15KDM4ECYP3A4TSHR
SCHEMBL29213350 0.78 GAA (0.49) GAAALOX15KDM4ECYP3A4TSHR
SCHEMBL29213354 0.78 GAA (0.49) GAAALOX15KDM4ECYP3A4TSHR
SCHEMBL30903305 0.78 GAA (0.49) GAAALOX15KDM4ECYP3A4TSHR
SCHEMBL11673049 0.78 ALDH1A1 (0.62) KDM4EALDH1A1TDP1MAPK1LDHA
SCHEMBL6237220 0.77 LDHA (0.57) RAB9AALDH1A1LDHA
SCHEMBL490932 0.77 LDHA (0.76) GAAALOX15KDM4ECYP3A4TSHR
SCHEMBL28049334 0.77 LDHA (0.57) RAB9AALDH1A1LDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011106114-A1 IDENTIFICATION OF HUMAN T2R RECEPTORS AND THE USE THEREOF TO IDENTIFY INHIBITORS (BLOCKERS) OF BITTER TASTE SENOMYX, INC. (US) 2011-09-01 WO disclosed
CN-1088083-A Cosmetic composition UNILEVER NV (NL) 1994-06-22 CN disclosed