SCHEMBL23840409

SCHEMBL23840409

COc1ncc(NC(=O)c2cnn(C)c2Cl)cc1S(=O)(=O)Nc1c(C)cccc1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 6/20 0.42
NR3C1 P04150 1/20 0.41
PIK3C3 Q8NEB9 1/20 0.40
IDH1 O75874 3/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 2/20 0.39
MEN1 O00255 2/20 0.39
LMNA P02545 2/20 0.39
KMT2A Q03164 2/20 0.39
MITF O75030 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
CHRNA7 P36544 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
BRAF P15056 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25487581 0.92 NPC1 (0.45) MALT1NR3C1PIK3C3KDM4EMEN1
SCHEMBL23840445 0.91 PIK3C3 (0.38) MALT1NR3C1PIK3C3KMT2AALDH1A1
SCHEMBL23840355 0.89 MALT1 (0.47) MALT1PIK3C3BRAF
SCHEMBL23840365 0.88 SMN1; SMN2 (0.41) MALT1PIK3C3MAPTKDM4EMEN1
SCHEMBL23840564 0.88 PIK3C3 (0.38) MALT1NR3C1PIK3C3MAPTKDM4E
SCHEMBL23840385 0.85 SMN1; SMN2 (0.48) NR3C1IDH1MAPTKDM4EMEN1
SCHEMBL25485494 0.85 KCNK3 (0.52) MAPTMEN1LMNAKMT2AALDH1A1
SCHEMBL23840544 0.84 ALDH1A1 (0.47) PIK3C3MAPTMEN1LMNAKMT2A
SCHEMBL23840341 0.84 KMT2A (0.46) PIK3C3MAPTKDM4EMEN1LMNA
SCHEMBL23840585 0.84 KDM4E (0.43) NR3C1PIK3C3IDH1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230159509-A1 PYRIDINESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-05-25 US disclosed
WO-2021188907-A1 PYRIDINESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2021-09-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230159509-A1 PYRIDINESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF TRAP1, PINK1, PPM1D MALT1 1352/4885NR3C1 2076/4885PIK3C3 1399/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.