SCHEMBL23846529

SCHEMBL23846529

COc1ccc(N)cc1S(=O)(=O)Nc1ccc(-c2ccccc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.60
LMNA P02545 2/20 0.60
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
ALOX12 P18054 1/20 0.60
BRD4 O60885 1/20 0.54
BRD2 P25440 1/20 0.54
BRD3 Q15059 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.52
HTT P42858 1/20 0.52
GAA P10253 1/20 0.52
ACLY P53396 4/20 0.52
WDR5 P61964 1/20 0.52
TRIM24 O15164 1/20 0.52
MAPT P10636 2/20 0.51
PIK3CD O00329 1/20 0.51
PIK3CA P42336 1/20 0.51
PIK3CG P48736 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23847019 0.92 MEN1 (0.61) ALPLLMNAMEN1KMT2AALOX12
SCHEMBL23846503 0.85 SMN1; SMN2 (0.71) ALPLLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL17980891 0.84 MAPT (0.60) ALPLLMNAMEN1KMT2AALOX12
SCHEMBL25754817 0.84 NPSR1 (0.62) ALPLLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL23846500 0.84 LMNA (0.73) ALPLLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL23847027 0.83 MEN1 (0.59) ALPLLMNAMEN1KMT2AALOX12
SCHEMBL23833758 0.81 RECQL (0.73) ALPLLMNASMN1; SMN2GAA
SCHEMBL23833737 0.81 MEN1 (0.63) ALPLLMNAMEN1KMT2AALOX12
SCHEMBL25754741 0.80 HPGD (0.57) ALPLLMNAMEN1KMT2AALOX12
SCHEMBL18385111 0.80 SMN1; SMN2 (0.60) LMNAMEN1KMT2AALOX12SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed
WO-2021188880-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2021-09-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF TRAP1, PINK1, TP53BP1 ALPL 3721/4885LMNA 3435/4885MEN1 3902/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.